Synthesis and Characterization of Novel 4-Methyl-3-isoxazolidinone Derivatives

Chemical Research in Chinese Universities ›› 2006, Vol. 22 ›› Issue (6): 717-720.doi:

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Synthesis and Characterization of Novel 4-Methyl-3-isoxazolidinone Derivatives

GAO Fei-fei¹, ZHANG Guang-liang¹, ZHENG Liang-yu², LI Yao-xian¹ and ZHANG Suo-qin¹

1. College of Chemistry,
2. Key Lab for Molecular Enzymology and Engineering, Ministry of Education, Jilin University, Changchun 130021, P. R. China

Received:2005-12-26 Revised:1900-01-01 Online:2006-11-25 Published:2006-11-25
Contact: ZHANG Suo-qin E-mail:zhangsq@jlu.edu.cn

Abstract

Abstract: A novel type of acetohydroxyacid synthase inhibitors, 4-methyl-3-isoxazolidinone derivatives of sulfonylurea, was designed and synthesized. The structures of these compounds were confirmed by using MS, NMR, and elemental analysis. The results of preliminary active tests indicate that the compounds show a herbicidal activity.

Key words: 4-Methyl-3-isoxazolidinone, Sulfonylureas, Acetohydroxyacid synthase, Herbicidal activity , 4-Methyl-3-isoxazolidinone, Sulfonylureas, Acetohydroxyacid synthase, Herbicidal activity

GAO Fei-fei , ZHANG Guang-liang , ZHENG Liang-yu , LI Yao-xian , ZHANG Suo-qin . Synthesis and Characterization of Novel 4-Methyl-3-isoxazolidinone Derivatives[J]. Chemical Research in Chinese Universities, 2006, 22(6): 717-720.

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Synthesis and Characterization of Novel 4-Methyl-3-isoxazolidinone Derivatives

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