Design and Synthesis of 3-(1-Phenylethyl)thiazolidine-2-thione Derivatives with Potential Biological Activities

高等学校化学研究 ›› 2011, Vol. 27 ›› Issue (3): 431-434.

Design and Synthesis of 3-(1-Phenylethyl)thiazolidine-2-thione Derivatives with Potential Biological Activities

LI Hong-xin, CHEN Xiao-tao and XU Liang-zhong*

College of Chemistry and Molecular Engineering, Qingdao University of Science and Technology, Qingdao 266042, P. R. China

收稿日期:2010-06-01 修回日期:2010-08-16 出版日期:2011-05-25 发布日期:2011-04-29
通讯作者: XU Liang-zhong E-mail:qknhs@yahoo.com.cn

Design and Synthesis of 3-(1-Phenylethyl)thiazolidine-2-thione Derivatives with Potential Biological Activities

LI Hong-xin, CHEN Xiao-tao and XU Liang-zhong*

College of Chemistry and Molecular Engineering, Qingdao University of Science and Technology, Qingdao 266042, P. R. China

Received:2010-06-01 Revised:2010-08-16 Online:2011-05-25 Published:2011-04-29
Contact: XU Liang-zhong E-mail:qknhs@yahoo.com.cn

摘要/Abstract

摘要： A series of novel neonicotinoids derivatives 4a―4p was designed and synthesized by introducing the ethylbenzene group into the thiazole ring, their structures were confirmed by IR, 1H NMR and elemental analysis. The crystal structure of compound 4j has been determined by X-ray diffraction analysis.

关键词: Crystal structure, Design, Neonicotinoids derivatives, Thiacloprid

Abstract: A series of novel neonicotinoids derivatives 4a―4p was designed and synthesized by introducing the ethylbenzene group into the thiazole ring, their structures were confirmed by IR, 1H NMR and elemental analysis. The crystal structure of compound 4j has been determined by X-ray diffraction analysis.

Key words: Crystal structure, Design, Neonicotinoids derivatives, Thiacloprid

LI Hong-xin, CHEN Xiao-tao and XU Liang-zhong*. Design and Synthesis of 3-(1-Phenylethyl)thiazolidine-2-thione Derivatives with Potential Biological Activities[J]. 高等学校化学研究, 2011, 27(3): 431-434.

LI Hong-xin, CHEN Xiao-tao and XU Liang-zhong*. Design and Synthesis of 3-(1-Phenylethyl)thiazolidine-2-thione Derivatives with Potential Biological Activities[J]. Chemical Research in Chinese Universities, 2011, 27(3): 431-434.

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Design and Synthesis of 3-(1-Phenylethyl)thiazolidine-2-thione Derivatives with Potential Biological Activities

Design and Synthesis of 3-(1-Phenylethyl)thiazolidine-2-thione Derivatives with Potential Biological Activities

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